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Title: Topical analgesic and
methods of use
United States Patent: 7,157,106
Issued: January 2, 2007
Inventors: Salmonson; Roger
S. (Westborough, MA)
Appl. No.: 10/608,744
Filed: June 27, 2003
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Abstract
Topical analgesics, generally comprising
calendula oil and cornmint oil, and methods of use.
SUMMARY OF THE
INVENTION
It is therefore a primary object of this
invention to provide a topical analgesic that reduces underlying pain when
applied directly to the skin.
It is a further object of this invention to provide a topical analgesic
that is particularly adapted to reduce pain associated with menstruation,
and more specifically to reduce menstrual cramping.
The analgesic and methods of the invention were developed as a result of
efforts to alleviate chronic pain via topical analgesics and more
specifically to develop a topical analgesic for temporary relief from
menstrual cramps. The analgesic obviates the need for individuals to
ingest systemic, unnecessary multi-symptom medication when the individual
is able to identify and topically target areas of bodily pain associated
with menstrual cramping.
A preferred formulation of the topical analgesic of the invention
generally comprises: 90% calendula oil mixed with 45% of one or more of
alcohol, mineral oil glycerin and water; and 10% cornmint oil.
Another preferred formulation of the topical analgesic of the invention
generally comprises: an effective amount of each of the following
components: cornmint oil; orange oil; pennyroyal oil; rosemary Spanish
oil; corianda oil; menthyl acetate; alpha pinene; beta pinene; camphor
white oil; calendula oil; mineral oil; and almond oil, wherein said
effective amounts are preferably about: 65 66% cornmint, 0.4 1.0% orange
oil; 4.0 5.0% pennyroyal oil; 6.0 7.0% rosemary Spanish oil; 0.2 0.4%
corianda oil; 1.0 2.0% menthyl acetate; 1.0 2.0% alpha pinene; 0.7 1.5%
beta pinene; 5.0 6.0% camphor white oil; 0.04 0.06% calendula oil; 0.02
0.03% mineral oil; and 15.0 16.0% almond oil.
Yet another preferred formulation of the topical analgesic of the
invention generally comprises: an effective amount of each of the
following components: cornmint oil, orange oil; pennyroyal oil; rosemary
Spanish oil; corianda oil; menthyl acetate; alpha pinene; beta pinene;
camphor white oil; calendula oil; and mineral oil, wherein said effective
amounts are preferably about: 80 81% cornmint oil, 0.4 1.0% orange oil;
4.0 5.0% pennyroyal oil; 6.0 7.0% rosemary Spanish oil; 0.2 0.4% corianda
oil; 1.0 2.0% menthyl acetate; 1.0 2.0% alpha pinene; 0.7 1.5% beta pinene;
5.0 6.0% camphor white oil; 0.04 0.06% calendula oil; and 0.02 0.03%
mineral oil.
A preferred formulation of the composition of the invention that is
particularly suited to reduce pain associated with menstruation,
comprising, 90% calendula oil mixed with 45% of one or more of alcohol,
mineral oil, glycerin or water; and 10% cornmint oil.
Another preferred formulation of the composition of the invention that is
particularly suited to reduce pain associated with menstruation,
comprising, an effective amount of each of the following components:
cornmint oil; orange oil; pennyroyal oil; rosemary Spanish oil; corianda
oil; menthyl acetate; alpha pinene; beta pinene; camphor white oil;
calendula oil; mineral oil; and almond oil, wherein said effective amounts
are preferably about: 65 66% cornmint, 0.4 1.0% orange oil; 4.0 5.0%
pennyroyal oil; 6.0 7.0% rosemary Spanish oil; 0.2 0.4% corianda oil; 1.0
2.0% menthyl acetate; 1.0 2.0% alpha pinene; 0.7 1.5% beta pinene; 5.0
6.0% camphor white oil; 0.04 0.06% calendula oil; 0.02 0.03% mineral oil;
and 15.0 16.0% almond oil.
Yet another preferred formulation of the composition of the invention that
is particularly suited to reduce pain associated with menstruation,
comprising, an effective amount of each of the following components:
cornmint oil, orange oil; pennyroyal oil; rosemary Spanish oil; corianda
oil; menthyl acetate; alpha pinene; beta pinene; camphor white oil;
calendula oil; and mineral oil, wherein said effective amounts are about:
80 81% cornmint oil, 0.4 1.0% orange oil; 4.0 5.0% pennyroyal oil; 6.0
7.0% rosemary Spanish oil; 0.2 0.4% corianda oil; 1.0 2.0% menthyl
acetate; 1.0 2.0% alpha pinene; 0.7 1.5% beta pinene; 5.0 6.0% camphor
white oil; 0.04 0.06% calendula oil; and 0.02 0.03% mineral oil.
Yet another preferred formulation of the composition that is particularly
suited to reduce pain associated with menstruation, comprising, an
effective amount of each of the following components: cornmint oil, orange
oil; pennyroyal oil; rosemary Spanish oil; corianda oil; menthyl acetate;
alpha pinene; beta pinene; camphor white oil; and calendula oil, wherein
said effective amounts are preferably about: 80 81% cornmint oil, 0.4 1.0%
orange oil; 4.0 5.0% pennyroyal oil; 6.0 7.0% rosemary Spanish oil; 0.2
0.4% corianda oil; 1.0 2.0% menthyl acetate; 1.0 2.0% alpha pinene; 0.7
1.5% beta pinene; 5.0 6.0% camphor white oil; and 0.04 0.06% calendula
oil.
A preferred method of the invention for reducing pain associated with
menstruation, comprising the steps of: providing a topical analgesic
comprising, an effective amount of calendula oil and an effective amount
of cornmint oil applying at least one coat of said analgesic directly on
skin over one or more areas of pain, wherein said step of applying
preferably comprises applying at least 3 4 coats directly on said skin
over one or more of said areas of pain; and keeping said areas of pain
warm for an effective amount of time. The topical analgesic used in the
method may further comprise, an effective amount of components selected
from a group consisting of: orange oil; pennyroyal oil; rosemary Spanish
oil; corianda oil; menthyl acetate; alpha pinene; beta pinene; camphor
white oil; calendula oil; mineral oil; and almond oil.
DETAILED DESCRIPTION
OF THE PREFERRED EMBODIMENTS AND METHODS
The topical analgesic of the invention is
intended for use as a general topical analgesic, but is especially suited
for reducing pain and discomfort associated with menstruation and
menstrual cramping. The analgesic and methods of the invention were
developed to alleviate chronic pain via topical analgesics and more
specifically to provide temporary relief from menstrual cramps. The
analgesic is topically applied to enable the individual to identify and
target the analgesic to areas where pain exists. As such, individuals do
not need to take unwanted and unnecessary multi-symptom oral medications
simply to alleviate menstrual cramping. This is particularly important in
view of the numerous, undesirable side effects associated with orally
administered painkillers. As an added benefit, the analgesic of the
invention comprises all naturally existing components.
There are several preferred formulations described herein but each of the
formulations comprise calendula oil and cornmint oil in varying
concentrations. The calendula oil is of particular active significance to
the formulation. Calendula oil has long been recognized as having possible
homeopathic uses such as facilitating skin abrasions and burns and as an
anti-inflammatory agent, antiseptic, astringent, cholagogue and
emmenagogue. However, we have discovered in our efforts to develop the
topical analgesic of the invention containing calendula oil has an
affirmative effect on nerve axions. Specifically, solutions of the
analgesic cause nerve cell axions to retreat. When the analgesic was
removed, the axional shape was restored.
Described below are several preferred formulations of the invention.
Formulation 1
90% calendula oil mixed with 45% of alcohol, mineral oil, glycerin and/or
oil; and
10% cornmint oil.
Formulation 2
An effective amount of each of the following: cornmint oil; orange oil;
pennyroyal oil; rosemary Spanish oil; corianda oil; menthyl acetate; alpha
pinene; beta pinene; camphor white oil; calendula oil; mineral oil; and
almond oil, wherein said effective amounts are preferably about:
65 66% cornmint,
0.4 1.0% orange oil;
4.0 5.0% pennyroyal oil;
6.0 7.0% rosemary Spanish oil;
0.2 0.4% corianda oil;
1.0 2.0% menthyl acetate;
1.0 2.0% alpha pinene;
0.7 1.5% beta pinene;
5.0 6.0% camphor white oil;
0.04 0.06% calendula oil;
0.02 0.03% mineral oil; and
15.0 16.0% almond oil.
Formulation 3
An effect amount of each of the following components: cornmint oil, orange
oil; pennyroyal oil; rosemary Spanish oil; corianda oil; menthyl acetate;
alpha pinene; beta pinene; camphor white oil; calendula oil; and mineral
oil, wherein said effective amounts are preferably about:
80 81% cornmint oil,
0.4 1.0% orange oil;
4.0 5.0% pennyroyal oil;
6.0 7.0% rosemary Spanish oil;
0.2 0.4% corianda oil;
1.0 2.0% menthyl acetate;
1.0 2.0% alpha pinene;
0.7 1.5% beta pinene;
5.0 6.0% camphor white oil;
0.04 0.06% calendula oil; and
0.02 0.03% mineral oil.
The preferred method of the invention for reducing pain, particularly pain
associated with menstruation, comprising the steps of: providing one or
more of the topical analgesics of any of the formulations described
herein, comprising, an effective amount of calendula oil and an effective
amount of cornmint oil; and applying at least one coat of the analgesic
directly on skin over one or more areas of pain, wherein said step of
applying preferably comprises applying at least 3 4 coats directly on said
skin over one or more of said areas of pain; and keeping said areas of
pain warm for an effective amount of time.
The analgesic is best applied using an applicator bottle that enables the
user to dispense small amounts of the analgesic to targeted areas of the
skin. For example, the applicator may comprise a roller ball or an
absorbent foam stopper. At the first sign of discomfort or pain, the
analgesic is applied directly to the skin over the area of discomfort or
pain by rubbing the applicator tip against the skin. The analgesic may be
gently massaged into the skin. Three to four coats are preferable,
although the effective amount may be varied as needed or desired. The area
of application should generally be about as large as the user's hand and
will remain moist on the skin for a few minutes after application. Relief
is typically obtained in less than ten to fifteen minutes after
application. Additional application may be necessary to achieve the
desired comfort level.
Although specific features of the invention are described in connection
with some of the formulations and methods and not others, this is for
convenience only as some feature may be combined with any or all of the
other features in accordance with the invention.
Claim 1 of 2 Claims
1. A composition adapted to reduce pain
associated with menstruation, comprising, an effective amount of each of
the following components: cornmint oil, orange oil; pennyroyal oil;
rosemary Spanish oil; corianda oil; menthyl acetate; alpha pinene; beta
pinene; camphor white oil; and calendula oil. ____________________________________________
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patent.
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